- Natural product: Cannabis (Cannabis sativa)
- Associated study: Cannabidiol, a major phytocannabinoid, as a potent atypical inhibitor for CYP2D6.
In Vitro Enzyme Inhibition Experiment
Recombinant: THC-dextramethorphan
Inhibition was detected. Cutoff used — Not specified
- CYP2D6 4173631
                                            Recombinant expression system  Baculovirus-insect cells
                                            
                                            
                                                
                                                Cytochrome B5  No
                                                
                                            
                                        
Results
Table 1
| Sample | Compound measured | Value | Measurement | Study sequence | Additional information | N replicates | 
|---|
Experimental Conditions
0.25 pmol
                                                            
                                                                Commercially available
                                                                
                                                                
                                                            
                                                        
200 μL
10 min
                                                            
                                                                MgCl2
                                                                
                                                                
                                                            
                                                                NADPH regenerating system
                                                                
                                                                
                                                            
                                                        
0.15-24 μM
5 min
                                                            
                                                                NADPH with precipitant
                                                                
                                                                
                                                            
                                                        
