OATP1A2 in vitro inhibition CSV JSON

In Vitro Transporter Inhibition Experiment

OATP1A2 in vitro inhibition

Inhibition was detected.  Cutoff used — not clearly specified

nadolol 1313200

(-)-epigallocatechin gallate

  • OATP1A2 (SLCO1A2)

Transfected / siRNA knock-out / injected cells HEK293 transfected cells

Results

Sample Compound measured Value Measurement Study sequence Additional information N replicates

Experimental Conditions

Cell Culture Conditions

poly-D-lysine hydrobromide-coated 12-well plates

2

Assay Conditions

5 min

37 deg C

7.3

100 µM

1, 10, 100, and 1000 µM

not specified