- Natural product: Cannabis (Cannabis sativa)
- Associated study: Characterization of major phytocannabinoids, cannabidiol and cannabinol, as isoform-selective and potent inhibitors of human CYP1 enzymes
In Vitro Enzyme Inhibition Experiment
HLMs: CBN
Inhibition was detected. Cutoff used — Not specified
- CYP1A1 4173297
Cell fraction Pooled human liver microsomes -7999662
Results
Tables 2 and 3.
IC50 at 20 min
Sample | Compound measured | Value | Measurement | Study sequence | Additional information | N replicates |
---|
Experimental Conditions
96-well
5 μg
Commercially available
200 μL
30 min
NADPH
150 nM
5 min
No NADPH with precipitant
0.025-25 μM