7-Hydroxymitragynine P-gp Inhibition CSV JSON

In Vitro Transporter Inhibition Experiment

7-Hydroxymitragynine P-gp Inhibition

Inhibition was detected.  Cutoff used —

EC50 positive control verapamil (22.3± 1.4 μM)

calcein-am

7-hydroxymitragynine

  • P-gp (ABCB1)

Transfected / siRNA knock-out / injected cells MDCK transfected cells

Results

positive control verapamil (22.3± 1.4 μM)

Fig 1S (with exact values in text pg 574)

Sample Compound measured Value Measurement Study sequence Additional information N replicates

Experimental Conditions

Cell Culture Conditions

70 000 cells/well

Assay Conditions

5 uM

5 uM

ChromaDex