In Vitro Enzyme Inhibition Experiment
Screening of kratom extracts as inhibitors CYP3A activity in HIM
Inhibition was detected. Cutoff used —
50% inhibition at the highest tested concentration
Cell fraction Pooled human intestinal microsomes -7999663
Three methanolic Kratom extracts were tested, K-50, K-51 and K-52.
|Sample||Compound measured||Value||Measurement||Study sequence||Additional information||N replicates|
2, 10, 20 µg/mL